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Ukubonisa 1-12 kweziphumo 29

CAS NO. IGAMA LEMVELISO AMAGQABANTSHINTSHI
    1527503-11-2 A-366 (1527503-11-2)

    I-366 yinto enamandla kwaye ikhetha i-G9a / GLP histone lysine methyltransferase inhibitor (IC₅₀ = 3.3 nM). Ibonisa> Ukukhethwa kwe-1000-fold for ...

    328968-36-1 I-C646 (328968-36-1)

    I-C646 inhibitor ye-histone acetyltransferase, kwaye inhibisa i-p300 nge-Ki ye-400 nM. Ukukhethwa ngokukhethekileyo kwe-p300 ngokubhekiselele kwezinye i-ace ...

    1163-36-6 I-Clemizole HCL (1163-36-6)

    I-Clemizole hydrochloride yi-H1 i-histamine i-receptor antagonist, ifumaneka ekuthintela ngokuphindaphindiweyo ukuphindaphinda kwe-HCV. IC50 yeClemizole ...

    1621862-70-1 I-CPI-1205 (1621862-70-1)

    I-CPI-1205 i-inhibitor ye-histone lysine methyltransferase ye-histone lysine methyltransferase ye-EZH2, enezinto ezinokuthi zenze i-antineoplastic.

    ...
    1396772-26-1 EPZ005687 (1396772-26-1)

    I-EPZ005687 iyisimo se-EZH2 esinamandla kunye nekhethi ye-24 nM, i-50-fold selectivity ngokumelene ne-EZH1 kunye ne-500-fold selectivity against 15 ...

    1616391-65-1 EPZ015666 (1616391-65-1)

    I-EPZ015666 inamandla, ikhetha i-PRMT5 inhibitor (i-Ki ye-5 nM); ubonisa> Ukukhethwa kwe-20,000 kwithuba kwezinye ii-PMTs. I-EPZ015666 isebenza nge-blocki ...

    1616391-87-7 EPZ015866 (GSK591) (1616391-87-7)

    I-EPZ015866 (GSK591) yiyona inhibitor ekhethileyo ye-arginine methyltransferase PRMT5 / MEP50 ubuncwane ngaloo ndlela ibeka i-methylation yayo ...

    1700663-41-7 EPZ020411 (1700663-41-7)

    I-EPZ020411 yindlela ekhuselekileyo yokukhetha i-PRMT6 kunye ne-IC50 ye-10 nM, ine> 10 ikhokhelo ye-PRMT6 ngaphezu kwe-PRMT1 kunye ne-PRMT8.

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    1380288-87-8 EPZ5676 (1380288-87-8)

    U-Pinometostat, owaziwa nangokuthi yi-EPZ-5676. I-Pinometostat isetyenziswe kwizilingo ekufundeni unyango lwe-Leukemia, i-Acute Leukemias, iMyeloid Acute ...

    1403254-99-8 EPZ6438 (1403254-99-8)

    I-Tazemetostat (EPZ-6438) yinto enamandla, ekhethiweyo kunye ngomlomo i-EZH2 inhibitor. UTazemetostat usetyenziswe kwizilingo ekufundeni unyango ...

    1373423-53-0 GSK J4 (1373423-53-0)

    I-GSK-J4 isetyenziselwe ukufunda isiphumo se-KDM2B (iJumonji (JmjC) domain history 3 i-lysine 36 (H3K36) i-di-demethylase) inhibition kusinda ...

    1431368-48-7 GSK-LSD1 2HCl (1431368-48-7)

    I-GSK-LSD1 isetyenziswe njenge-lysine ethile ye-demethylase i-1 (LSD1) inhibitor kwimigundane yokufunda ukufelwa kwe-sepsis. Kuye kwasetyenziswa ...